Arimidex (Anastrozole) CAS:120511-73-1

Description

By blocking the aromatase enzyme, Arimidex directly lowers the levels of estrogen circulating in the body. This is critical for treating breast cancer because of estrogen's function on cancer cells. Still, it also serves a great purpose for steroid users, as estrogen is the enemy of steroid use and is responsible for many of the severe side effects we all want to avoid.

As one of the best aromatase inhibitors, Arimidex is considered the most effective choice for combating the estrogenic side effects of aromatizing steroid use like gynecomastia, water retention, and the associated high blood pressure that can come with excess water retention.

While not all steroids aromatize, the most common anabolic steroids that you're likely to be using, like all forms of Testosterone, Nandrolone, Dianabol, and others, come with strong estrogenic effects as a result of aromatization.

Therefore, the use of Arimidex in post-cycle therapy is going to be a high priority for the majority of steroid users, whether you're a beginner, an advanced user, or somewhere in between.

Clinical Data

Is Arimidex a good estrogen blocker?

Yes, Arimidex (anastrozole) is considered an effective estrogen blocker, specifically an aromatase inhibitor. As mentioned earlier, it works by inhibiting the enzyme aromatase, which is responsible for the conversion of other hormones (such as androgens) into estrogen. By blocking this process, Arimidex reduces the overall levels of estrogen in the body, particularly in postmenopausal women.

In the context of breast cancer treatment, Arimidex is commonly used to suppress estrogen production in hormone receptor-positive (HR+) breast cancer, where the cancer cells depend on estrogen for growth and proliferation. By lowering estrogen levels, Arimidex helps to slow down or inhibit the growth of HR+ breast cancer tumors.

Aromatase inhibitors like Arimidex are often preferred over other estrogen-blocking medications, such as tamoxifen, in postmenopausal women with HR+ breast cancer because they are more effective in reducing estrogen levels. However, the choice of treatment depends on several factors, including the stage and type of breast cancer, the patient's medical history, and individual health considerations.

It is crucial for patients to work closely with their oncologist or healthcare provider to determine the most appropriate treatment plan, considering potential side effects and overall benefits of using Arimidex or any other medication.

Arimidex Dosage

Anastrozole Dosage During Anabolic Steroid Use

Arimidex is a highly effective aromatase inhibitor at low doses for estrogen control when using steroids that aromatize. Many guys will find that 0.5mg every two days is enough to mitigate all side effects.

Others will need to increase to 1mg every two days. While some people will take as much as 1mg of Arimidex every day during a cycle, this is usually unnecessary, and it's also advised to test your individual response to the drug by starting out at the lower dose.

Female Arimidex Dosage

Because it has such strong estrogen suppressive effects, Arimidex is mostly only given to post-menopausal women as a breast cancer treatment to slow the growth of some types of tumors and where the cancer is still progressing after the use of SERM drugs. The most common dosage is 1mg daily.

Many women will be required to take Arimidex for up to five years to help control the growth of cancerous tumors. This long-term administration of Arimidex comes with an increased risk of side effects that we rarely or never see with the short-term use that steroid users undertake with this drug.

As Arimidex is not prescribed medically for the majority of women with breast cancer who have not yet reached menopause, female steroid users also should not use this drug for any purpose.

Arimidex Dosage for PCT and Increased Endogenous Testosterone Secretion

As mentioned already, Arimidex is not a prime choice for post-cycle therapy purposes for the majority of steroid users.

While it has some function for helping stimulate the production of testosterone, its highly suppressive effects on estrogen can result in a less-than-ideal effect on testosterone production and a result that is not as effective as using SERMs like Nolvadex and Clomid, which are more commonly used for PCT purposes, in conjunction with hCG (Human chorionic gonadotropin).

While everyone reacts differently to different drugs, and your post-cycle therapy will also depend on the type of steroid cycle you were on, some may wish to include Arimidex. A dosage of 0.5mg to 1mg daily during the post-cycle therapy cycle is sufficient in these cases.

Arimidex vs. Nolvadex for PCT

More and more bodybuilders are turning to AIs like Arimidex to meet their needs for a powerful and effective anti-estrogen while using steroids because AIs actually block the function of estrogen. At the same time, SERMs like Nolvadex are very selective in how and where they can stop the functioning of estrogen. But many of us are still using Nolvadex and other SERMs, often in conjunction with AIs.

How does Nolvadex compare with Arimidex, and should you still be using a SERM at all? It's not so black and white, and ultimately, it comes down to how your body reacts to the drugs, the strength of your steroid cycle, and the associated side effects.

A big advantage that Nolvadex and other SERMs have over Arimidex and AIs is that while Arimidex is likely to have a negative impact on your cholesterol by lowering HDL cholesterol – the good cholesterol type and this is amplified further when it's used with most anabolic steroids, Nolvadex does not come with this concern.

In fact, Nolvadex can potentially be good for cholesterol, quite the opposite of Arimidex in this regard. This is a big reason, especially for those concerned with cholesterol health, that people will choose to use SERMs over an AI like Arimidex, particularly for more mild steroid cycles where an AI might not be needed anyway.

There's another huge benefit to Nolvadex, though: it is very effective during post-cycle therapy to stimulate the natural production of testosterone following suppression during a steroid cycle.

Arimidex and SERMs, in general, don't excel at this function because although it has some testosterone-stimulating effects, the way Arimidex suppresses estrogen levels so much that there is not enough for normal functioning makes testosterone stimulation relatively weak and not often enough to provide the much-needed benefits during post cycle therapy.

Therefore, Arimidex is rarely recommended for use during post-cycle therapy and instead is considered to be a drug that is mainly used during a steroid cycle, which is where its performance and results do outshine that of Nolvadex.

That's not to say that bodybuilders don't use Arimidex during post-cycle therapy: many do, but only in conjunction with other drugs so that every possible angle is covered to aid in total recovery from a powerful steroid cycle.

For people foregoing Arimidex altogether during post-cycle therapy, a combination of Clomid, Nolvadex, and hCG is often used instead.

The ultimate goal of post-cycle therapy is to stimulate testosterone not only for normal functioning as a male but also to retain your muscle gains and control body fat – both of which will suffer when testosterone levels are lower than normal.

Important Safety Information About ARIMIDEX

Prescription ARIMIDEX is only for postmenopausal women. ARIMIDEX should not be taken if you are pregnant because it may harm your unborn child. Do not take ARIMIDEX if you are allergic to any of its ingredients

Based on information from a study in patients with early breast cancer, women with a history of blockages in heart arteries (ischemic heart disease) who take ARIMIDEX may have a slight increase in this type of heart disease compared to similar patients who take tamoxifen

ARIMIDEX can cause bone softening/weakening (osteoporosis) increasing the chance of fractures. In a clinical study in early breast cancer, there were more fractures (including fractures of the spine, hip, and wrist) with ARIMIDEX (10%) than with tamoxifen (7%)

In a clinical study in early breast cancer, some patients taking ARIMIDEX had an increase in cholesterol. Skin reactions, allergic reactions, and changes in blood tests of liver function have also been reported

In the early breast cancer clinical trial, the most common side effects seen with ARIMIDEX include hot flashes, joint symptoms (including arthritis and arthralgia), weakness, mood changes, pain, back pain, sore throat, nausea and vomiting, rash, depression, high blood pressure, osteoporosis, fractures, swelling of arms/legs, insomnia, and headache

In advanced breast cancer trials, the most common side effects seen with ARIMIDEX versus tamoxifen include hot flashes, nausea, decreased energy and weakness, pain, back pain, headache, bone pain, increased cough, shortness of breath, sore throat, and swelling of arms and legs. Joint pain/stiffness has been reported in association with the use of ARIMIDEX

ARIMIDEX should not be taken with tamoxifen or estrogen-containing therapies

Approved Uses for ARIMIDEX

ARIMIDEX is approved for adjuvant treatment (treatment following surgery with or without radiation) of postmenopausal women with hormone receptor-positive early breast cancer.

ARIMIDEX is approved for the initial treatment of postmenopausal women with hormone receptor-positive or hormone receptor-unknown locally advanced or metastatic breast cancer and for the treatment of postmenopausal women with advanced breast cancer that has progressed following treatment with tamoxifen. Patients with hormone receptor-negative disease and patients who did not previously respond to tamoxifen therapy rarely responded to ARIMIDEX.

Our Advantages

1.Quality:every item is strictly tested by our professional staff and get ISO certificate.
2.Price: much lower than our peers since we are factory. A discount would be given when you make a large order.
3.Delivery: We have adequate stock so we can make the delivery within 24 hours after payment.
4.Perfect Reshipping policy has been made to protect customers max bennefits and reduce the potentical losses.
5.Good after-sale service: always keeping track on the status of your parcel until delivered and trying our utmost to solve customers problems entounered
6.main products:Raw steroids,human growth hormone,Semi-finished oils,bodybuilding peptides,SARMs raws,Anabolic steroids