Toremifene Citrate( Fareston ) CAS:89778-27-8

Description

Toremifene (also known under its brand and trade name of Fareston) is a member of a category, family, and class of drugs that are known as SERMs (Selective Estrogen Receptor Modulators). SERMs fall under an even broader category of drugs that are known as anti-estrogens, and the cousin family of SERMs (that also fall under anti-estrogens) are aromatase inhibitors, commonly abbreviated as AIs. SERMs include compounds such as Toremifene, Nolvadex (Tamoxifen), and Clomid (Clomiphene Citrate). Aromatase inhibitors (AIs) include compounds such as Arimidex (Anastrozole), Aromasin (Exemestane), and Letrozole (Femara). Although the two fall under the category of anti-estrogens, they are both sub-categories that branch off into their own families, as SERMs and AIs differ greatly in their mechanism of action within the human body concerning how they control or block Estrogen.

Toremifene Citrate (Fareston, Acapodene) is an oral selective estrogen receptor modulator (SERM) which helps oppose the actions of estrogen in the body. Chemically related to tamoxifen, toremifene is a selective estrogen receptor modulator (SERM). This agent binds competitively to estrogen receptors, thereby interfering with estrogen activity. Toremifene also has intrinsic estrogenic properties, which are manifested according to tissue type or species.

Fareston (toremifene citrate) is an estrogen agonist/antagonist that blocks estrogen from reaching cancer cells used to slow the growth of metastatic breast cancer (cancer that has spread from the original tumor). Unlike chemotherapy, Fareston does not actually destroy cancer cells.

Clinical Data

Fareston Benefits (Toremifene Effects)

As a SERM drug, Fareston is not a performance-enhancement substance but is one that is considered a useful ancillary drug for some steroid users.

Fareston has some clear benefits for anabolic steroid users. Most importantly, it is highly useful in your efforts to combat estrogenic side effects that are caused by many steroids. These include the development of gyno, as well as water retention and increased blood pressure. The growth of male breast tissue, called gynecomastia is the main use of Fareston. It is made to target breast tissue receptors so it is here specifically we see its greatest benefit.

Users can make use of Fareston to prevent gyno symptoms from occurring or to reduce and eliminate gyno signs if they've started occurring while using aromatizing steroids.

High dosages of steroids and males who are particularly sensitive to gyno development are likely also to need the addition of an aromatase inhibitor drug (AI) to mitigate gynecomastia. The negative impact of some AIs on cholesterol should be considered, though, with Fareston, by comparison, actually having some potential cholesterol benefits as described below.

When it comes to other estrogenic side effects like water retention and the associated increase in blood pressure it can bring about, Fareston may not always provide enough benefit to combat these issues completely in users who are either using highly aromatizing steroids, using these steroids at very high doses, and who have a less than ideal diet.

In more moderate steroid cycles and where the diet is kept lower in carbohydrates, it can be possible to control water retention well by using Fareston and without the addition of other drugs.

An unexpected benefit of this medication is its effect on cholesterol due to its function in the liver. Many anabolic steroids have a negative impact on cholesterol levels, causing great concern to users.

Fareston may be able to help mitigate this risk somewhat by improving lipid profiles so that LDL, or bad cholesterol levels, are reduced while encouraging the increase in HDL or good cholesterol levels. Many steroids have the opposite effect on cholesterol, making this a particularly useful drug for those steroid users who are concerned about their cholesterol health during a cycle.

Another benefit that Fareston has when compared with Nolvadex is that Fareston is not known to negatively impact IGF-1. This makes it much more suitable to use during a steroid cycle when you do not want to see your IGF-1 levels decrease. While Fareston is a younger drug than Nolvadex, and this same effect might still yet be found in the future, for now, it is strongly believed that Fareston does not exhibit the same negative impact on IGF-1 levels when used for estrogen mitigation during a steroid cycle.

Fareston may have other health benefits over other SERMs like Nolvadex. Early studies show that Fareston is likely to tax the liver less than Nolvadex. While this isn't a huge concern for short-term use, if you plan on using any SERM on a regular basis, liver health is critical to consider – particularly as many steroids can stress the liver.

There are certainly pros and cons to using Fareston. The positive benefits and effects are appealing to anyone wanting to focus specifically on preventing gyno. This is where Toremifene delivers the greatest benefit, rather than in the PCT stage where, as yet, it is not showing to be as strong a choice as Nolvadex.

Is Toremifene The Same As Tamoxifen?

Toremifene and tamoxifen are similar but distinct medications belonging to the same class of drugs known as selective estrogen receptor modulators (SERMs). They share some similarities in their mechanism of action and usage but also have differences.

Both medications work by blocking the effects of estrogen in certain tissues. They are used in the treatment of breast cancer, particularly in hormone receptor-positive breast cancers where the cancer cells depend on estrogen to grow.

Here are some differences between toremifene and tamoxifen:

1. Chemical Structure: While they both fall under the SERM class, they have different chemical structures. Toremifene is a chlorinated derivative of tamoxifen.

2. FDA Approval: Tamoxifen has been approved for both early and advanced breast cancer, as well as for reducing the risk of breast cancer in high-risk women. Toremifene is specifically approved for treating metastatic breast cancer in postmenopausal women.

3. Metabolism: They are metabolized differently in the body, potentially resulting in varied side effects and interactions with other medications.

4. Effectiveness and Side Effects: While both drugs have similarities in their efficacy against breast cancer, they may have different side effect profiles. Some individuals may tolerate one drug better than the other.

Both drugs are prescribed by healthcare providers based on individual patient needs, considering factors like the stage of cancer, medical history, and potential side effects.

How to take Toremifene Citrate

Oral routeMedicines used to treat cancer are very strong and can have many side effects. Before receiving this medicine, make sure you understand all the risks and benefits. It is important for you to work closely with your doctor during your treatment.

Your doctor will tell you how much medicine to use. Do not use more than directed.

Missed dose: Take a dose as soon as you remember. If it is almost time for your next dose, wait until then and take a regular dose. Do not take extra medicine to make up for a missed dose.

Store the medicine in a closed container at room temperature, away from heat, moisture, and direct light.

Store the medicine in a closed container at room temperature, away from heat, moisture, and direct light.

Oral routeMedicines used to treat cancer are very strong and can have many side effects. Before receiving this medicine, make sure you understand all the risks and benefits. It is important for you to work closely with your doctor during your treatment.

Missed dose: Take a dose as soon as you remember. If it is almost time for your next dose, wait until then and take a regular dose. Do not take extra medicine to make up for a missed dose.

Your doctor will tell you how much medicine to use. Do not use more than directed.

What to do if you miss a dose of Toremifene Citrate

Take a dose as soon as you remember. If it is almost time for your next dose, wait until then and take a regular dose. Do not take extra medicine to make up for a missed dose.

Keep all medicine out of the reach of children. Never share your medicine with anyone.

Oral routeAsk your pharmacist, doctor, or health caregiver about the best way to dispose of any leftover medicine after you have finished your treatment. You will also need to throw away old medicine after the expiration date has passed.

Our Advantages

1.Quality:every item is strictly tested by our professional staff and get ISO certificate.
2.Price: much lower than our peers since we are factory. A discount would be given when you make a large order.
3.Delivery: We have adequate stock so we can make the delivery within 24 hours after payment.
4.Perfect Reshipping policy has been made to protect customers max bennefits and reduce the potentical losses.
5.Good after-sale service: always keeping track on the status of your parcel until delivered and trying our utmost to solve customers problems entounered
6.main products:Raw steroids,human growth hormone,Semi-finished oils,bodybuilding peptides,SARMs raws,Anabolic steroids